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Canadian Pharmacist Qualifying Exam Practice · Question

What is the primary therapeutic target for direct oral anticoagulants (DOACs) like rivaroxaban or apixaban?

DOACs like rivaroxaban and apixaban directly inhibit Factor Xa, while dabigatran directly inhibits thrombin. This mechanism distinguishes them from warfarin, wh

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Question: What is the primary therapeutic target for direct oral anticoagulants (DOACs) like rivaroxaban or apixaban?

Answer options: ✅ Factor Xa or thrombin

  • Vitamin K epoxide reductase
  • Platelet aggregation
  • Prothrombin time (PT)

Correct answer: Factor Xa or thrombin

Explanation: DOACs like rivaroxaban and apixaban directly inhibit Factor Xa, while dabigatran directly inhibits thrombin. This mechanism distinguishes them from warfarin, which inhibits vitamin K epoxide reductase.

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