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Canadian Pharmacist Qualifying Exam Practice · Question

What is the primary mechanism of action of metformin in type 2 diabetes?

Metformin primarily works by decreasing hepatic glucose production and improving insulin sensitivity in peripheral tissues. It does not stimulate insulin secret

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Question: What is the primary mechanism of action of metformin in type 2 diabetes?

Answer options:

  • Stimulates insulin secretion from pancreatic beta cells
  • Increases glucose uptake by peripheral tissues ✅ Decreases hepatic glucose production
  • Inhibits alpha-glucosidase enzymes in the intestine

Correct answer: Decreases hepatic glucose production

Explanation: Metformin primarily works by decreasing hepatic glucose production and improving insulin sensitivity in peripheral tissues. It does not stimulate insulin secretion directly.

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