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Canadian Pharmacist Qualifying Exam Practice · Question

What is the primary mechanism by which sildenafil (Viagra) treats erectile dysfunction?

Sildenafil is a PDE5 inhibitor, which increases cyclic guanosine monophosphate (cGMP) levels in the corpus cavernosum, leading to smooth muscle relaxation and i

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Question: What is the primary mechanism by which sildenafil (Viagra) treats erectile dysfunction?

Answer options: ✅ Inhibiting phosphodiesterase-5 (PDE5) to increase cGMP levels.

  • Directly stimulating nitric oxide release.
  • Blocking alpha-adrenergic receptors.
  • Increasing testosterone production.

Correct answer: Inhibiting phosphodiesterase-5 (PDE5) to increase cGMP levels.

Explanation: Sildenafil is a PDE5 inhibitor, which increases cyclic guanosine monophosphate (cGMP) levels in the corpus cavernosum, leading to smooth muscle relaxation and increased blood flow.

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