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Canadian Pharmacist Qualifying Exam Practice · Question

Which antiplatelet medication irreversibly inhibits cyclooxygenase-1 (COX-1) in platelets?

Acetylsalicylic acid (ASA) is a cornerstone antiplatelet therapy that works by irreversibly inhibiting COX-1, preventing thromboxane A2 synthesis.

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Question: Which antiplatelet medication irreversibly inhibits cyclooxygenase-1 (COX-1) in platelets?

Answer options:

  • Clopidogrel
  • Ticagrelor ✅ Acetylsalicylic acid (ASA)
  • Dipyridamole

Correct answer: Acetylsalicylic acid (ASA)

Explanation: Acetylsalicylic acid (ASA) is a cornerstone antiplatelet therapy that works by irreversibly inhibiting COX-1, preventing thromboxane A2 synthesis.

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