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Canadian Pharmacist Qualifying Exam Practice · Question

What is the primary role of naloxone in opioid overdose?

Naloxone is a pure opioid antagonist that rapidly reverses the effects of opioid overdose, particularly respiratory depression, by displacing opioids from their

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Question: What is the primary role of naloxone in opioid overdose?

Answer options:

  • To increase opioid metabolism
  • To act as a partial opioid agonist ✅ To reverse opioid-induced respiratory depression
  • To prevent opioid cravings

Correct answer: To reverse opioid-induced respiratory depression

Explanation: Naloxone is a pure opioid antagonist that rapidly reverses the effects of opioid overdose, particularly respiratory depression, by displacing opioids from their receptors.

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