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Canadian Pharmacist Qualifying Exam Practice · Question

Which drug is contraindicated in patients with a history of angioedema related to ACE inhibitor use?

Lisinopril is an ACE inhibitor, and its use is contraindicated in patients with a history of angioedema related to any ACE inhibitor due to cross-reactivity.

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Question: Which drug is contraindicated in patients with a history of angioedema related to ACE inhibitor use?

Answer options:

  • Valsartan (an ARB) ✅ Lisinopril (an ACE inhibitor)
  • Amlodipine (a CCB)
  • Metoprolol (a beta-blocker)

Correct answer: Lisinopril (an ACE inhibitor)

Explanation: Lisinopril is an ACE inhibitor, and its use is contraindicated in patients with a history of angioedema related to any ACE inhibitor due to cross-reactivity.

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