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Canadian Pharmacist Qualifying Exam Practice · Question

What is the primary mechanism of action of sacubitril/valsartan in heart failure?

Sacubitril/valsartan is an angiotensin receptor-neprilysin inhibitor (ARNI) that improves outcomes in heart failure by blocking angiotensin II effects and incre

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Question: What is the primary mechanism of action of sacubitril/valsartan in heart failure?

Answer options: ✅ Angiotensin receptor and neprilysin inhibition

  • Beta-adrenergic receptor blockade
  • Direct renin inhibition
  • Sodium-glucose cotransporter 2 inhibition

Correct answer: Angiotensin receptor and neprilysin inhibition

Explanation: Sacubitril/valsartan is an angiotensin receptor-neprilysin inhibitor (ARNI) that improves outcomes in heart failure by blocking angiotensin II effects and increasing natriuretic peptides.

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