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Canadian Pharmacist Qualifying Exam Practice · Question

What is the primary mechanism of action of ACE inhibitors in managing hypertension?

ACE inhibitors block the conversion of angiotensin I to angiotensin II, leading to vasodilation, reduced aldosterone secretion, and decreased blood pressure.

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Question: What is the primary mechanism of action of ACE inhibitors in managing hypertension?

Answer options: ✅ Inhibition of angiotensin-converting enzyme, leading to reduced angiotensin II and aldosterone.

  • Blocking of beta-adrenergic receptors, reducing heart rate and cardiac output.
  • Direct relaxation of vascular smooth muscle, causing vasodilation.
  • Increased excretion of sodium and water by the kidneys.

Correct answer: Inhibition of angiotensin-converting enzyme, leading to reduced angiotensin II and aldosterone.

Explanation: ACE inhibitors block the conversion of angiotensin I to angiotensin II, leading to vasodilation, reduced aldosterone secretion, and decreased blood pressure.

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